{"id":1355,"date":"2026-02-24T10:25:10","date_gmt":"2026-02-24T10:25:10","guid":{"rendered":"https:\/\/www.almacgroup.com\/discovery\/?page_id=1355"},"modified":"2026-02-24T10:29:50","modified_gmt":"2026-02-24T10:29:50","slug":"science","status":"publish","type":"page","link":"https:\/\/www.almacgroup.com\/discovery\/science\/","title":{"rendered":"Science"},"content":{"rendered":"\n<p> <\/p>\n\n\n\n<h1 class=\"wp-block-heading\" id=\"h-science\">Science<\/h1>\n\n\n\n<h2 class=\"wp-block-heading\" id=\"h-for-almost-two-decades-almac-discovery-has-been-innovating-across-therapeutic-targets-disease-indications-and-targeting-modalities\">For almost two decades Almac Discovery has been innovating across therapeutic targets, disease indications and targeting modalities.\u00a0<\/h2>\n\n\n\n<p><strong>We have built deep internal expertise and collaborative networks that have enabled us to deliver scientific programs that fully align with our commitment to develop life-changing treatments for patients<\/strong><\/p>\n\n\n\n<p>Building on our success in developing novel small molecules targeting kinases (e.g. WEE1 \u2013 Ph1b, AKT \u2013 Ph3), small domain antibody drug conjugates (ADCs) and being recognised as the leader in deubiquitinase drug discovery, our current strategy leverages our deep integrated expertise to deliver next generation ADCs featuring novel payloads and linker technologies. Additionally, we are harnessing induced proximity to develop molecules targeting emerging disease relevant proteins that can be developed either as novel payloads for new ADCs or as novel oral therapeutics.<\/p>\n\n\n\n<figure class=\"wp-block-image size-large\"><img decoding=\"async\" width=\"1024\" height=\"425\" data-src=\"https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/almac-discovery-science-infographic-1024x425.png\" alt=\"\" class=\"wp-image-1356 lazyload\" data-srcset=\"https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/almac-discovery-science-infographic-1024x425.png 1024w, https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/almac-discovery-science-infographic-300x124.png 300w, https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/almac-discovery-science-infographic-768x318.png 768w, https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/almac-discovery-science-infographic-1536x637.png 1536w, https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/almac-discovery-science-infographic-1351x560.png 1351w, https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/almac-discovery-science-infographic-480x199.png 480w, https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/almac-discovery-science-infographic.png 1710w\" data-sizes=\"(max-width: 1024px) 100vw, 1024px\" src=\"data:image\/gif;base64,R0lGODlhAQABAAAAACH5BAEKAAEALAAAAAABAAEAAAICTAEAOw==\" style=\"--smush-placeholder-width: 1024px; --smush-placeholder-aspect-ratio: 1024\/425;\" \/><noscript><img decoding=\"async\" width=\"1024\" height=\"425\" src=\"https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/almac-discovery-science-infographic-1024x425.png\" alt=\"\" class=\"wp-image-1356\" srcset=\"https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/almac-discovery-science-infographic-1024x425.png 1024w, https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/almac-discovery-science-infographic-300x124.png 300w, https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/almac-discovery-science-infographic-768x318.png 768w, https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/almac-discovery-science-infographic-1536x637.png 1536w, https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/almac-discovery-science-infographic-1351x560.png 1351w, https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/almac-discovery-science-infographic-480x199.png 480w, https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/almac-discovery-science-infographic.png 1710w\" sizes=\"(max-width: 1024px) 100vw, 1024px\" \/><\/noscript><\/figure>\n\n\n\n<div style=\"height:100px\" aria-hidden=\"true\" class=\"wp-block-spacer\"><\/div>\n\n\n\n<h3 class=\"wp-block-heading\" id=\"h-almac-discovery-s-adc-approach-is-designed-to-optimize-both-therapeutic-performance-and-development-efficiency-by-integrating-several-key-features\">Almac Discovery\u2019s ADC approach is designed to optimize both therapeutic performance and development efficiency by integrating several key features:<br><\/h3>\n\n\n<!-- thirds_media_text.php -->\n<!-- Two thirds text, One third Media -->\n<section class=\"u-bg-white t-theme-component-overwrite\"  id=\"thirdsMediaBlock\">\n\t<div class=\"c-half-media-text\">\n\t\t<div class=\"o-wrapper\">\n\t\t\t\n\t\t\t\t\t\n\t\t\t\t\t\t<article class=\"o-grid \">\n\t\t\t\t\t\t\t<div class=\"u-width-2\/3 u-width-full@m c-half-media__repeat-text none u-bg-white\">\n\t\t\t\t\t\t\t\t\t\t\t\t\t\t\t\t<ul>\n<li>The use of a <strong>smaller antibody format <\/strong>enhances tumour penetration, enabling more effective delivery of the cytotoxic payload to cancer cells<\/li>\n<li><strong>Bispecific binding <\/strong>further strengthens this approach by improving target engagement, which can increase efficacy while maintaining a favourable safety profile<\/li>\n<li>Payload attachment through <strong>engineered linkages <\/strong>supports improved manufacturability, helping to ensure consistent production and scalability of the ADC platform.<\/li>\n<li><strong>Novel payloads <\/strong>beyond traditional chemotherapeutics is a core strategy for the development of new ADCs<\/li>\n<\/ul>\n\t\t\t\t\t\t\t\t\t\t\t\t\t\t\t<\/div>\n\t\t\t\t\t\t\t<div class=\"u-width-1\/3 u-width-full@m c-half-media__repeat-image\">\n\t\t\t\t                <!-- \n-->\n\n\n\t\t\t\t\t\t\t\t\t<img decoding=\"async\" data-src=\"https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/image-2.png\" alt=\"\" src=\"data:image\/gif;base64,R0lGODlhAQABAAAAACH5BAEKAAEALAAAAAABAAEAAAICTAEAOw==\" class=\"lazyload\" style=\"--smush-placeholder-width: 1920px; --smush-placeholder-aspect-ratio: 1920\/1080;\"><noscript><img decoding=\"async\" src=\"https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/image-2.png\" alt=\"\"><\/noscript>\n\t\t\t\t                \t\t\t\t\t\t\t<\/div>\n\t\t\t\t\t\t<\/article>\n\n\t\t\t\t\t\n\t\t\t\t\t<\/div>\n\t<\/div>\n<\/section>\n\n\n\n<div style=\"height:100px\" aria-hidden=\"true\" class=\"wp-block-spacer\"><\/div>\n\n\n\n<h3 class=\"wp-block-heading\" id=\"h-we-apply-computation-and-chemistry-driven-strategies-to-advance-the-development-of-novel-molecular-degraders-mgds-and-innovative-small-molecule-inhibitors-both-as-standalone-therapeutics-and-as-antibody-drug-conjugate-adc-payloads-innovative-chemistry-is-essential-for-next-generation-mg-discovery-this-approach-is-underpinned-by\">We apply computation and chemistry\u2011driven strategies to advance the development of novel molecular degraders (MGDs) and innovative small molecule inhibitors, both as standalone therapeutics and as antibody\u2013drug conjugate (ADC) payloads. Innovative chemistry is essential for next\u2011generation MG discovery. This approach is underpinned by:<\/h3>\n\n\n<!-- thirds_media_text.php -->\n<!-- Two thirds text, One third Media -->\n<section class=\"u-bg-white t-theme-component-overwrite\"  id=\"thirdsMediaBlock\">\n\t<div class=\"c-half-media-text\">\n\t\t<div class=\"o-wrapper\">\n\t\t\t\n\t\t\t\t\t\n\t\t\t\t\t\t<article class=\"o-grid \">\n\t\t\t\t\t\t\t<div class=\"u-width-2\/3 u-width-full@m c-half-media__repeat-text none u-bg-white\">\n\t\t\t\t\t\t\t\t\t\t\t\t\t\t\t\t<ul>\n<li aria-level=\"1\">Continual expansion of MGD screening libraries based on <b>novel scaffolds <\/b>and innovative chemistries<\/li>\n<li aria-level=\"1\">Integration of <b>computational chemistry and AI\/ML\u2011based methods <\/b>to enable efficient target identification and rational compound design<\/li>\n<li aria-level=\"1\"><b>Strategic collaborations <\/b>that accelerate new molecular glue discovery (e.g. Northern Ireland Chemoproteomics Centre-of-Excellence)<\/li>\n<\/ul>\n\t\t\t\t\t\t\t\t\t\t\t\t\t\t\t<\/div>\n\t\t\t\t\t\t\t<div class=\"u-width-1\/3 u-width-full@m c-half-media__repeat-image\">\n\t\t\t\t                <!-- \n-->\n\n\n\t\t\t\t\t\t\t\t\t<img decoding=\"async\" data-src=\"https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/image-3-e1771859321581.png\" alt=\"\" src=\"data:image\/gif;base64,R0lGODlhAQABAAAAACH5BAEKAAEALAAAAAABAAEAAAICTAEAOw==\" class=\"lazyload\" style=\"--smush-placeholder-width: 200px; --smush-placeholder-aspect-ratio: 200\/187;\"><noscript><img decoding=\"async\" src=\"https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/image-3-e1771859321581.png\" alt=\"\"><\/noscript>\n\t\t\t\t                \t\t\t\t\t\t\t<\/div>\n\t\t\t\t\t\t<\/article>\n\n\t\t\t\t\t\n\t\t\t\t\t<\/div>\n\t<\/div>\n<\/section>\n\n\n\n<div style=\"height:100px\" aria-hidden=\"true\" class=\"wp-block-spacer\"><\/div>\n\n\n\n<p>We have developed a global network of life sciences contract research organizations (CROs) and strategic partners, strengthened by deep industry\u2013academia collaborations that drive innovative and translational R&amp;D. Key partnerships include the Future Medicines Institute (FMI) and the NI Chemoproteomics Centre of Excellence, enabling access to cutting-edge scientific expertise, advanced technologies, and collaborative research models to accelerate the discovery and development of future medicines.<\/p>\n\n\n\n<div class=\"wp-block-columns is-layout-flex wp-container-core-columns-is-layout-9d6595d7 wp-block-columns-is-layout-flex\">\n<div class=\"wp-block-column is-layout-flow wp-block-column-is-layout-flow\">\n<figure class=\"wp-block-image size-full\"><a href=\"https:\/\/www.futuremedicinesinstitute.com\/ \"><img decoding=\"async\" width=\"756\" height=\"334\" data-src=\"https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/image-5.png\" alt=\"\" class=\"wp-image-1366 lazyload\" data-srcset=\"https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/image-5.png 756w, https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/image-5-300x133.png 300w, https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/image-5-480x212.png 480w\" data-sizes=\"(max-width: 756px) 100vw, 756px\" src=\"data:image\/gif;base64,R0lGODlhAQABAAAAACH5BAEKAAEALAAAAAABAAEAAAICTAEAOw==\" style=\"--smush-placeholder-width: 756px; --smush-placeholder-aspect-ratio: 756\/334;\" \/><noscript><img decoding=\"async\" width=\"756\" height=\"334\" src=\"https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/image-5.png\" alt=\"\" class=\"wp-image-1366\" srcset=\"https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/image-5.png 756w, https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/image-5-300x133.png 300w, https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/image-5-480x212.png 480w\" sizes=\"(max-width: 756px) 100vw, 756px\" \/><\/noscript><\/a><\/figure>\n<\/div>\n\n\n\n<div class=\"wp-block-column is-layout-flow wp-block-column-is-layout-flow\">\n<figure class=\"wp-block-image size-full\"><a href=\"https:\/\/gtr.ukri.org\/projects?ref=BB\/Y00325X\/1 \"><img decoding=\"async\" width=\"476\" height=\"248\" data-src=\"https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/image-4.png\" alt=\"\" class=\"wp-image-1365 lazyload\" data-srcset=\"https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/image-4.png 476w, https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/image-4-300x156.png 300w\" data-sizes=\"(max-width: 476px) 100vw, 476px\" src=\"data:image\/gif;base64,R0lGODlhAQABAAAAACH5BAEKAAEALAAAAAABAAEAAAICTAEAOw==\" style=\"--smush-placeholder-width: 476px; --smush-placeholder-aspect-ratio: 476\/248;\" \/><noscript><img decoding=\"async\" width=\"476\" height=\"248\" src=\"https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/image-4.png\" alt=\"\" class=\"wp-image-1365\" srcset=\"https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/image-4.png 476w, https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/image-4-300x156.png 300w\" sizes=\"(max-width: 476px) 100vw, 476px\" \/><\/noscript><\/a><\/figure>\n<\/div>\n<\/div>\n","protected":false},"excerpt":{"rendered":"<p>Science For almost two decades Almac Discovery has been innovating across therapeutic targets, disease indications and targeting modalities.\u00a0 We have built deep internal expertise and collaborative networks that have enabled us to deliver scientific programs that fully align with our commitment to develop life-changing treatments for patients Building on our success in developing novel small [&hellip;]<\/p>\n","protected":false},"author":2229,"featured_media":0,"parent":0,"menu_order":0,"comment_status":"closed","ping_status":"closed","template":"template-article-publication.php","meta":{"_acf_changed":false,"footnotes":""},"class_list":["post-1355","page","type-page","status-publish","hentry"],"acf":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO Premium plugin v25.3.1 (Yoast SEO v26.3) - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>Science - Discovery<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/www.almacgroup.com\/discovery\/science\/\" \/>\n<meta property=\"og:locale\" content=\"en_GB\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Science\" \/>\n<meta property=\"og:description\" content=\"Science For almost two decades Almac Discovery has been innovating across therapeutic targets, disease indications and targeting modalities.\u00a0 We have built deep internal expertise and collaborative networks that have enabled us to deliver scientific programs that fully align with our commitment to develop life-changing treatments for patients Building on our success in developing novel small [&hellip;]\" \/>\n<meta property=\"og:url\" content=\"https:\/\/www.almacgroup.com\/discovery\/science\/\" \/>\n<meta property=\"og:site_name\" content=\"Discovery\" \/>\n<meta property=\"article:modified_time\" content=\"2026-02-24T10:29:50+00:00\" \/>\n<meta property=\"og:image\" content=\"https:\/\/www.almacgroup.com\/discovery\/wp-content\/uploads\/sites\/2\/2026\/02\/almac-discovery-science-infographic.png\" \/>\n\t<meta property=\"og:image:width\" content=\"1710\" \/>\n\t<meta property=\"og:image:height\" content=\"709\" \/>\n\t<meta property=\"og:image:type\" content=\"image\/png\" \/>\n<meta name=\"twitter:card\" content=\"summary_large_image\" \/>\n<meta name=\"twitter:label1\" content=\"Estimated reading time\" \/>\n\t<meta name=\"twitter:data1\" content=\"2 minutes\" \/>\n<script type=\"application\/ld+json\" class=\"yoast-schema-graph\">{\"@context\":\"https:\/\/schema.org\",\"@graph\":[{\"@type\":\"WebPage\",\"@id\":\"https:\/\/www.almacgroup.com\/discovery\/science\/\",\"url\":\"https:\/\/www.almacgroup.com\/discovery\/science\/\",\"name\":\"Science - 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